鲁拉西酮

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鲁拉西酮

鲁拉西酮

编号ABP001018 化学名称Lurasidone CAS367514-87-2 分子式C28H36N4O2S 分子量492.676 纯度 98%

化学名称 : 鲁拉西酮

CAS : 367514-87-2

英文名称: Lurasidone

英文同义词: (3aR,4S,7R,7aS)-2-[[(1R,2R)-2-[[4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl]methyl]cyclohexyl]methyl]hexahydro-4,7-methano-1H-isoindole-1,3(2H)-dione

生物活性

Potent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types. Centrally active following oral administration.
询价