化学名称 : SB 525334/SB525334
CAS : 356559-20-1
英文名称: SB 525334/SB525334
英文同义词: 6-[2-(1,1-Dimethylethyl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-4-yl]quinoxaline
溶解度:DMSO
储存条件:at -20°
生物活性
SB525334 is a selective inhibitor of transforming growth factor-β receptor I (ALK5, TGF-βRI) (IC50=14.3 nM). This agent inhibits TGF-β-induced ALK5 serine/ threonine kinase activity, thereby preventing phosphorylation of the Smad transcription factors and subsequent gene activation.参考文献
[1] Laping NJ. IDrugs 1999;2:907-14