ESI-09

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ESI-09

ESI-09

Cat.No.ABP027301 Chemical NameESI-09 CAS263707-16-0 MolFormula MolWeight Purity NLT 98%

Chemical Name : ESI-09

CAS : 263707-16-0

ESI-09 is a novel noncyclic nucleotide EPAC antagonist that is capable of specifically blocking intracellular EPAC-mediated Rap1 activation and Akt phosphorylation, as well as EPAC-mediated insulin secretion in pancreatic β cells with IC50 of 1.4 uM/3.2 uM for EPAC2/EPAC1 respectively.
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