PIK75/PIK-75 hydrochloride

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PIK75/PIK-75 hydrochloride

PIK75/PIK-75 hydrochloride

Cat.No.ABP000105 Chemical NamePIK75/PIK-75 hydrochloride CAS945619-31-8 MolFormulaC16H15BrClN5O4S MolWeight488.743 Purity >99%

Chemical Name : PIK75/PIK-75 hydrochloride

CAS : 945619-31-8

Synonyms: N'-[(1E)-(6-Bromoimidazo[1,2-A]pyridin-3-yl)methylene]-N,2-dimethyl-5-nitrobenzenesulfonohydrazide hydrochloride


Storage:-20C 2 years


PI3K p110α specific inhibitor; IC50 values (nM): 7.8 (p110α), 343 (p110β), 907 (p110δ) (Chaussade et al reported).


ZA Knight et al. A Pharmacological Map of the PI3-K Family Defines a Role for p110α in Insulin Signaling. Cell 2006, 125, 733–747.


C Chaussade et al. Evidence for functional redundancy of class IA PI3K isoforms in insulin signalling. Biochem J. 2007, 404(3), 449–458.