183288-99-5

RJR 2403 oxalate

183288-99-5

Cat.No.ABP000370 Chemical NameRJR 2403 oxalate MolFormulaC12H16N2O4 MolWeight252.2664 Purity >99 %

Chemical Name : RJR 2403 oxalate

CAS : 183288-99-5

Synonyms: (E)-N-Methyl-4-(3-pyridinyl)-3-bute n-1-amine oxalate

Solubility:Soluble to 100 mM in water

Storage:Desiccate at +4°C

Biologieal

A neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki values are 26 and 36000 nM for α4β2 and α7 receptors respectively). Active in vivo

Reference

Bencherif et al (1996) RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J.Pharmacol.Exp.Ther.

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